Detailed clinical resources and information regarding Anticancer Therapies.

Hormonal Therapies

Estrogen Endocrine Therapy
GnRH agonistGoserelin (Zoladex) – Leuprolide (Eligard, Lupron, Viadur) – Triptorelin (Decapeptyl)
AI (steroidal)Exemestane (Aromasin)
AI (non-steroidal)Anastrozole (Arimidex) – Letrozole (Femara)
Selective ER modulators (SERMs)Raloxifene (Evista) – Tamoxifen (Nolvadex) – Toremifene (Fareston)
Selective ER down regulators (SERDs)Elacestrant (Orserdu) – Fulvestrant (Faslodex) – Imlunestrant (Inluriyo) – Camizestrant (investigational) – Vepdegestrant (PROTAC ER degrader, investigational)
Androgen Deprivation Therapy (ADT)
GnRH agonistBuserelin (Suprefact) – Goserelin (Zoladex®) – Histrelin (Supprelin LA®, Vantas®) – Leuprolide (Eligard®, Lupron®) – Triptorelin (Trelstar®)
GnRH antagonistDegarelix (Firmagon®)
Androgen Hormonal Therapy
Antiandrogen (steroidal)Cyproterone acetate
Antiandrogen (non-steroidal) (-amide)Apalutamide (Erleada) – Bicalutamide (Casodex) – Darolutamide (Nubeqa) – Enzalutamide (Xtandi) – Flutamide (Eulexin) – Nilutamide (Nildandron)
CYP17 (Androgen biosynthesis) inhibitorAbiraterone acetate (Zytiga) – Ketoconazole (n/a)
Somatostatin Analog
 Lanreotide (Somatuline Depot) – Octreotide (Bynfezia; Mycapssa; SandoSTATIN)

Chemotherapy

Alkylating Agents
Nitrogen mustardsBendamustine (Treanda, Bendeka) – Chlorambucil (Leukeran) – CycloPHOSphamide (Cytoxan, Neosar) – Ifosfamide (Ifex) – Mechlorethamine (Topical for CTCL; Valchlor) – Melphalan (Alkeran, Evomela) – Melphalan flufenamide (Pepaxto; withdrawn 2022)
NitrosureasCarmustine (BiCNU, Gliadel Wafer [brain tumors]) – Lomustine (CeeNU, Gleostine) – Streptozocin (Zanosar)
Platinum analogsCISplatin (Platinol) – CARBOplatin (Paraplatin) – Oxaliplatin (Eloxatin)
TriazenesDacarbazine (DTIC-Dome) – Temozolomide (Temodar)
Alkyl SulfonatesBusulfan (Myleran PO, Busulfex IV) – Treosulfan
EthyleneiminesThiotepa (Tepadina)
MethylmelamineAltretamine (Hexalen)
Methylhydrazine derivativeProcarbazine (Matulane)
Marine-derived / minor groove bindersTrabectedin (Yondelis), Lurbinectedin (Zepzelca for SCLC)
Antimetabolite Agents (CCS – S-Phase)
Fluoropyrimidines5-Fluorouracil (Adrucil) – Capecitabine (Xeloda PO) – Floxuridine HAI – Trifluridine + Tipiracil (Lonsurf)
Cytidine Analogs (C)Azacitidine (Vidaza) – Cytarabine (Conventional, Cytosar-U; Liposomal+Daunorubicin, Vyxeos) – Decitabine (Dacogen) – Gemcitabine (Gemzar)
Purines and Purine AntimetabolitesCladribine (Leustatin) – Clofarabine (Clolar) – Fludarabine (Fludara) – Mercaptopurine (6-MP, Purinethol, Purixan PO) – Nelarabine (Arranon) – Pentostatin (Nipent) – Thioguanine (6-TG, Tabloid)
AntifolatesMethotrexate (Trexall, Rheumatrex, Otrexup, Rasuvo) – PEMEtrexed (Alimta) – PRALAtrexate (Folotyn) – Raltitrexed (Tomudex)
Ribonucleoside diphosphate reductase inhHydroxyurea (Droxia; Hydrea; Siklos)  
Microtubule-Targeting Agents (CCS – M-Phase)
Vinca alkaloidsVinBLAStine (Velban) – VinCRIStine (Oncovin) – Vindesine (Eldisine) – Vinorelbine (Navelbine)
TaxanesCabazitaxel (Jevtana) – DOCEtaxel (Taxotere) – PACLitaxel (Conventional; Taxol) – PACLitaxel (Protein Bound; nab-paclitaxel, Abraxane)
HalichondrinsEribulin (Halaven)
Epothilone B analogIxabepilone (Ixempra)
Estradiol, nitrogen mustard, anti-microtubuleEstramustine (Emcyt)
ADC (microtubule-targeting warhead)Brentuximab Vedotin (BV; Adcetris; antiCD30) – Mirvetuximab Soravtansine (MIRV; Elahere; Anti-FRα) – Ado-Trastuzumab Emtansine (T-DM1; Kadcyla; antiHER2) – Enfortumab Vedotin-ejfv (EV; Padcev; Anti-Nectin-4) – Tisotumab Vedotin-tftv (TV; Tivdak; Anti-TF)
Cytotoxic Antibiotics
DNA break, ROS genBleomycin (BLEO 15K)
DNA intercalation / RNA polymerase inhibitionDACTINomycin (Actinomycin D; Cosmegen)
Bioreductive alkylationMitoMYcin C (Mutamycin)
Topoisomerase Inhibitors
(TopoI) Campothecin analogsIrinotecan (Camptosar) – Topotecan (Hycamtin)
(TopoII) EpipodophyllotoxinEtoposide (Vepesid) – Etoposide phosphate (Etopophos) – Teniposide (Vumon)
(TopoII) AnthracyclinesDAUNOrubicin (Conventional) – DOXOrubicin (Conventional; Adriamycin) – DOXOrubicin (Liposomal) – EpiRUBicinIDArubicinMitoXANTRONE (Novantrone) – Valrubicin (Valstar)
(TopoI) ADC Anti-Trop-2 warheadSacituzumab Govitecan (Trodelvy), Datopotamab Deruxtecan (Datroway)
Protein Synthesis Inhibitors
Cephalotaxine alkaloid (elongation inhibitor)Omacetaxine (Synribo)
Enzymes
 Asparaginase (Erwinia [Recombinant]) (Rylaze) – Calaspargase Pegol (Asparlas) – Pegaspargase (Oncaspar)

Targeted Therapy

EGFR Inhibitors
Monoclonal antibodiesCetuximab (Erbitux) – Necitumumab (Portazza) – Panitumumab (Vectibix)
First generation (reversible TKI)Erlotinib (Tarceva) – Gefitinib (Iressa)
Second-Generation (irreversible EGFR/HER2 TKIs)Afatinib (Gilotrif) – Dacomitinib (Vizimpro) – Lapatinib (Tykerb) –Neratinib (Nerlynx) – Vandetanib (Caprelsa)
Third-Generation (mutant-selective irreversible TKIs, T790M)Lazertinib (Leclaza) – Osimertinib (Tagrisso)
EGFR Exon 20 Insertions TKIMobocertinib (Exkivity) – Sunvozertinib (Zegfrovy)
KRAS G12C-inhibitorsAdagrasib (Krazati) – Sotorasib (Lumakras) – Olomorasib (investigational)
Bispecific mAb EGFR/MET Exon 20Amivantamab-vmjw (Rybrevant)
Human Epidermal Growth Factor Receptor 2 (HER2, ERBB2 GENE, P185) Antagonists
Monoclonal antibodiesTrastuzumab (Herceptin) – Ado-trastuzumab ematansine (Kadcyla) – Fam-trastuzumab deruxtecan-nxki (Enhertu) – Pertuzumab (Pertaja) – Zanidatamab-hrii (Ziihera)
Small moleculesLapatinib (Tykerb) – Neratinib (Nerlynx) – Tucatinib (Tukysa) – Zongertinib (Hernexeos)
HER2/HER3 bispecific inh mAbZenocutuzumab (Bizengri)
Claudin 18.2 (CLDN18.2) Inhibitor
Monoclonal antibodiesZolbetuximab-clzb (Vyloy)
Anaplastic Lymphoma Kinase (ALK) Inhibitors
First generationCrizotinib (Xalkori)
Second generationAlectinib (Alecensa) – Brigatinib (Alunbrig) – Ceritinib (Zykadia)
Third generationLorlatinib (Lorbrena)
ALK/ROS1 inhibitorTaletrectinib (Ibtrozi) – Entrectinib (Rozlytrek)
Neurotrophic tyrosine receptor kinase (NTRK) Inhibitors
TrkA, TrkB, TrkC inhibitorLarotrectinib (Vitrakvi)
Dual NTRK/ROS1 inhibitorEntrectinib (Rozlytrek) – Repotrectinib (Augtyro)
BRAF Inhibitors
TKI inhibitorsDabrafenib (Tafinlar) – Encorafenib (Braftovi) – Vemurafenib (Zelboraf) – Tovorafenib (Ojemda)
Mitogen-activated protein kinase (MEK) Inhibitors
KI inhibitorsBinimetinib (Mektovi) – Cobimetinib (Cotellic) – Mirdametinib (Gomekli) – Selumetinib (Koselugo) – Trametinib (Mekinist)
RAF/MEK, FAK/Pyk2i, RAF/MEKAvutometinib (novel RAF/MEK clamp) + Defactinib (FAK/Pyk2i) (Avmapki Fakzynja)
Mammalian Target Of Rapamycin (mTOR) Inhibitors
RapalogsEverolimus (Afinitor) – SirolimusTemsirolimus (Torisel)
Dual pan-PI3K/mTORC1/2iGedatolisib (investigational)
Phosphatidylinositol 3-Kinase (PI3K) Inhibitors
(α) Small moleculeAlpelisib (Piqray) – Inavolisib (Itovebi)
(α/δ) Small moleculeCopanlisib (Aliqopa)
(δ/γ) Small moleculeDuvelisib (Copiktra)
(δ) Small moleculeIdelalisib (Zydelig)
(δ/ε) Small moleculeUmbralisib (Ukoniq)
Dual pan-PI3K/mTORC1/2iGedatolisib (investigational)
Proteasome Inhibitors (PI)
First generationBortezomib (Velcade)
Second generationCarfilzomib (Kyprolis), Ixazomib (Ninlaro)
AKT Inhibitors
TKI inhibitorsCapivasertib (Truqap)
Vascular Endothelial Growth Factor (VEGF) Inhibitors
Monoclonal antibodies (-mab)Bevacizumab (Avastin) – Ramucirumab (Cyramza)
Recombinant fusion protein (-cept)Ziv-aflibercept (Zaltrap)
Small molecules (target TKI; -nib)Axitinib (Inlyta) – Cabozantinib (Cabometyx, Cometriq) – Fruquintinib (Fruzaqla) – Lenvatinib (Lenvima) – Pazopanib (Votrient) – Regorafenib (Stivarga; targets RAF TKI) – Sorafenib (Nexavar) – Suntinib (Sutent) – Tivozanib (Fotivda) – Vandetanib (Capresla)
MET Inhibitors
TKI inhibitorsCapmatinib (Tabrecta) – Crizotinib (Xalkori) – Tepotinib (Tepmetko)
Bispecific mAb EGFR/MET Exon 20Amivantamab-vmjw (Rybrevant)
ADC anti-cMet mAbTelisotuzumab Vedotin (Emrelis)
Fibroblast Growth Factor Receptor (FGFR) Inhibitors
mAb, HER2, GEJBemarituzumab (investigational)
TKI inhibitorErdafitinib (Balversa) – Futibatinib (Lytgobi) – Infigratinib (Truseltiq) – Pemigatinib (Pemazyre)
RET Kinase Inhibitors
TKI inhibitorPralsetinib (Gavreto) – Selpercatinib (Retevmo)
PDGFR-Alpha Blocker
Monoclonal antibodyOlaratumab (Lartruvo)
Small molecules, TKI inhibitorsAvapritinib (Ayvakit) – Ripretinib (Qinlock; KIT inhibitor)  
CDK 4/6 Inhibitors
Small moleculeAbemaciclib (Verzenio®) – Palbociclib (Ibrance®) – Ribociclib (Kisqali®)
Aurora A Kinase (AURKA) Inhibitors
Reversible, ATP-competitive, selectiveAlisertib (investigational)
BCL2 Inhibitors
 Venetoclax (Venclexta)
Poly (ADP-ribose) Polymerase (PARP) Inhibitors
TKI inhibitorsNiraparib (Zejula) – Olaparib (Lynparza) – Rucaparib (Rubraca) – Talazoparib tosylate (Talzenna)
BCR-ABL Inhibitors
First-generation TKIImatinib (Gleevec)
Second generation TKIDasatinib (Sprycel) – Nilotinib (Tasigna) – Bosutinib (Bosulif)
Third generation TKIPONATinib (Iclusig; T315I mutation)
TKI-STAMP inhibitorAsciminib (Scemblix)
Bruton Tyrosine Kinase (BTK) Inhibitors
1st gen TKI (covalent/irreversible)Ibrutinib (Imbruvica)
2nd gen TKI (covalent/irreversible)Acalabrutinib (Calquence) – Zanubrutinib (Brukinsa) – Tirabrutinib (Velexbru, investigational) – Orelabrutinib (Hibruka, Yinuokai, investigational)
3rd gen TKI (noncovalent)Pirtobrutinib (Jaypirca)
Dual BTK/LYNi (noncovalent)Birelentinib (investigational)
Janus Kinase (JAK) Inhibitors
Selective JAK2i TKIVGT1849B (investigational)
Dual JAK1/2 TKIMomelotinib (Ojjaara) – Ruxolitinib (Jakavi)
Dual FLT3/JAK2iFedratinib (Inrebic) – Pacritinib (Vonjo)
FLT3 Inhibitors
Class I (ITD-/TKD-mutations)Gilteritinib (Xospata) – Midostaurin (Rydapt)
Class II (ITD-mutations)Quizartinib (Vanflyta)
Dual FLT3/JAK2iFedratinib (Inrebic) – Pacritinib (Vonjo)
CSF-1R Inhibitors
Monoclonal antibodyAxatilimab-csfr (Niktimvo)
TKI inhibitorsPexidartinib (Turalio) – Vimseltinib (Romvimza)
Histone Deacetylase (HDAC) Inhibitors
 Belinostat (Beleodaq) – Panobinostat (Farydak) – RomiDEPsin (Istodax) – Vorinostat (Zolinza)
Histone Methyltransferase (HMT) Inhibitors
EZH2 inhibitorTazemetostat (Tazverik)
Menin Inhibitors
Menin-KMT2A interaction inhibitorRevumenib (Revuforj)
IDH1 Inhibitors
 Ivosidenib (Tibsovo) – Olutasidenib (Rezlidhia)
IDH2 Inhibitors
 Enasidenib (IDHIFA)
IDH1/2 Inhibitors
 Vorasidenib (Voranigo)
Selective Inhibitor Of Nuclear Export (SINE)
 Selinexor (Xpovio)
Gamma Secretase Inhibitors
 Nirogacestat (Ogsiveo)
Ornithine Decarboxylase Inhibitors
 Eflornithine (Iwilfin)
Glutaminase Inhibitors
 Telaglenastat (investigational)
Hepcidin Mimetic Peptides (Iron Regulators)
 Rusfertide (investigational)
HIF-2alpha Inhibitors
 Belzutifan (Welireg)
Hedgehog Pathway Inhibitors
 Glasdegib (Daurismo) – Sonidegib (Odomzo) – Vismodegib (Erivedge)
Telomerase Inhibitors
 Imetelstat (Rytelo) – Ateganosine (2′‑Deoxythioguanosine, investigational)
Selective Immunomodulating Microtubule-Binding Agent (SIMBA)
 Plinabulin (investigational)
Protease Activator Therapies (Oncogenic Stress Modulators)
 Dordaviprone (Modeyso)
Targeted Protein Modification
Degrader (PROTAC)Vepdegestrant (SERDs, investigational)
Rewires (RIPTAC)HLD-0915 (investigational)

Immunotherapy

Immune Checkpoint Inhibitors (ICI; CTLA-4, PD-1, PD-L1)
CTLA-4 inhibitorsIpilimumab (Yervoy®) – Tremelimumab-actl (Imjudo)
PD-1 inhibitorsCemiplimab-rwlc (Libtayo®) – Dostarlimab-gxly (Jemperli) – Nivolumab (Opdivo®) – Pembrolizumab (Keytruda) – Pembrolizumab and Berahyaluronidase (Keytruda Qlex) – Penpulimab (Anniko) – Retifanlimab (Zynyz) – Tislelizumab-jsgr (Tevimbra) – Toripalimab (Loqtorzi)
PD-L1 inhibitorsAtezolizumab (Tecentriq®) – Avelumab (Bavencio®) – Cosibelimab (Unloxcyt) – Durvalumab (Imfinzi®)
Dual LAG-3i/PD-1iNivolumab and Relatlimab (Opdualag)
CD47i fusion proteinEvorpacept (ALX148, investigational)
Bispecific PD-1/VEGFiIvonescimab (investigational)
Bispecific PD-L1/VEGFiPumitamig (investigational)
Anti-TIGIT Antibody
 Ociperlimab (investigational)
Bispecific T-Cell Engager (BiTE) Therapy
Anti-BCMA/CD3; mAbElranatamab (Elrexfio) – Teclistamab-cqyv (Tecvayli) – Linvoseltamab (Lynozyfic) – Alnuctamab (Investigational)
Anti-CD19/CD3; mAbBlinatumomab (Blincyto)
Anti-CD20/CD3; mAbEpcoritamab (Tepkinly) – Glofitamab (Columvi) – Mosunetuzumab (Lunsumio) – Cevostamab (investigational) – Odronextamab (investigational)
Anti-GPRC5D/CD3; mAbTalquetamab (Talvey)
Anti-gp100/CD3; rfp recombinant fusion proteinTebentafusp (Kimmtrak)
Anti-Delta-like ligand 3 (DLL3)/CD3; mAbTarlatamab (Imdelltra)
Trispecific T-Cell Engager (TRiTE) Therapy (investigational)
CD3, CD19, CD28CC312 (ongoing trial)
CD3, CD38, CD28SAR442257 (ongoing trial)
CD3, BCMA, CD38ISB-2001 (ongoing trial)
CD3, DLL3, albuminMK-6070 (formerly HPN328; ongoing trial)
CD3, BCMA, albuminHPN217 (ongoing trial)
CD3, EpCAM, blockHPN601 (ongoing trial)
CD3, CD79b, CD20JNJ-8543 (ongoing trial)
CD3, BCMA, GPRC5DJNJ-5322 (ongoing trial)
CD3, CD19, CD22AZD5492 (ongoing trial)
CD3, DLL3, PDL1ZG006 (ongoing trial)
Anti-CD19
mAbTafasitamab-cxix (Minjuvi)
Anti-CD20
mAbIbritumomab Tiuxetan (Zevalin) – Obinutuzumab (Gazyva) – Ofatumumab (Arzerra) – RiTUXimab (Rituxan, MabThera)
Anti-CD22
mAbMoxetumomab pasudotox-tdfk (Lumoxiti)
Anti-CD38
mAbDaratumumab (Darzalex, Darzalex Faspro as SC combo with hyaluronidase) – Isatuximab-irfc (Sarclisa)
Anti-CD52
mAbAlemtuzumab (Campath, Lemtrada)
Anti-SLAMF7
mAbElotuzumab (Empliciti)
Anti-GD2
mAbDinutuximab (Ch14.18; Unituxin) and Dinutuximab beta (Qarziba) – Naxitamab (Danyelza)
Anti-CC Chemokine Receptor 4 (CCR4) Antibody
mAbMogamulizumab-kpkc (Poteligeo)
Antibody-Drug Conjugate (ADC)
Anti-BCMABelantamab Mafodotin-blmf (Blenrep; withdrawn as it did not meet primary endpoint in DREAMM-3 PhIII)
Anti-B7-H3 (CD276)Ifinatamab Deruxtecan (I-DXd, investigational)
Anti-CD19Loncastuximab Tesirine-lpyl (Zynlonta)
Anti-CD22Inotuzumab Ozogamicin (Besponsa)
Anti-CD30Brentuximab Vedotin (Adcetris)
Anti-CD33Gemtuzumab Ozogamicin (Mylotarg)
Anti-CD79BPolatuzumab Vedotin (Polivy)
Anti-CDH177MW4911 (investigational)
Anti-cMetTelisotuzumab Vedotin (Emrelis)
Anti-Folate Receptor αMirvetuximab Soravtansine (Elahere) – Rinatabart Sesutecan (Rina-S, investigational)
Anti-HER2Ado-Trastuzumab Emtansine (Kadcyla) – Fam-Trastuzumab Deruxtecan (Enhertu) – Trastuzumab pamirtecan (BNT323, investigational)
Anti-Nectin-4Enfortumab Vedotin (Padcev)
Anti-Tissue FactorTisotumab Vedotin-tftv (Tivdak)
Anti-Trop-2Sacituzumab Govitecan (Trodelvy), Datopotamab Deruxtecan (Datroway)
Bispecific (EGFR x HER3)Izalontamab Brengitecan (Iza-bren, investigational)
Peptide-Drug Conjugate (PDC)
Anti-SORT1PQ203 (investigational)    
Cellular Therapies
CAR-T BCMACiltacabtagene autoleucel (Cilta-cel, Carvykti) – Idecabtagene vicleucel (Abecma)
CAR-T CD19Tisagenlecleucel (Kymriah) – Axicabtagene ciloleucel (Yescarta) – Brexucabtagene autoleucel (Tecartus) – Lisocabtagene maraleucel (Breyanzi) – Obecabtagene autoleucel (Aucatzyl)
CAR-T EGFRCARv3-TEAM-E
Tumor-Infiltrating Lymphocyte (TIL)Lifileucel (Amtagvi)
TCR MAGE-A4 antigenAfamitresgene Autoleucel (Tecelra; C-144-01 study)
VaccineSipuleucel-T
Gene TherapyAtidarsagene Autotemcel (Lenmeldy) – Betibeglogene Autotemcel (Zynteglo) – Elivaldogene Autotemcel (Skysona) – Exagamglogene Autotemcel (Casgevy) – Lovotibeglogene Autotemcel (Lyfgenia)
Immunomodulators
Small moleculeLenalidomide (Revlimid) – Pomalidomide (Pomalyst) – Thalidomide (Thalomid)  
Biological Response Modulators
IL-2Aldesleukin (Proleukin)
IL-15Nogapendekin Alfa Inbakicept (Anktiva, Adstiladrin)
VaccineBCG (Intravesical) (TICE BCG)
Interferon/PegsInterferon Alfa-2b (Intron A) – Peginterferon Alfa-2a (Pegasys) – Peginterferon Alfa-2b (Pegintron D/C) – Ropeginterferon Alfa-2b (Besremi)
IL2/CD25iDenileukin Diftitox
Anti-CD123Tagraxofusp (Elzonris)
Mannan-binding lectin-Associated Serine Protease-2 (MASP-2) Inhibitor – (Complement Modulation)
mAb complement inhNarsoplimab (investigational)
Oncolytic Virus
Genetically engineeredTalimogene Laherparepvec (T-VEC, Imlygic)
Stem-cell loaded viral txCLD-201 (SuperNova; investigational)

Genetic Therapy

Gene Therapy (Biologic Response Modifier)
human interferon alpha 2B (IFNα2b)Nadofaragene firadenovec-vncg (Adstiladrin®)

Differentiation Therapy

Arsenic Derivative
 Arsenic trioxide (Trisenox)
Retinoids
Retinoic Acid DerivativeAlitretinoin (Panretin) – Bexarotene (Targretin) – Isotretinoin (Absorica; Accutane; Amnesteem; Claravis; Clarus; Epuris; Myorisan [DSC]; Zenatane) – Tretinoin (ATRA, Vesanoid)
Retinoid-Like CompoundAcitretin (Soriatane)

Radiopharmaceutical

??[ZA1] 
 Radium-223 (??)

Supportive Therapy

RANK Ligand Inhibitors (Bone Health)
 Denosumab (Prolia, Xgeva)
Bisphosphonate (Bone Health)
 Alendronate (Binosto, Fosamax) – Clodronate (Clasteon) – Ibandronate (Boniva) – Pamidronate (Aredia) – Risedronate (Actonel; Atelvia) – Zoledronic Acid (Reclast, Aclasta, Zometa)
Hypoxia-Inducible Factor (HIF) Modulators (Anemia)
 Roxadustat (Evrenzo)